GBR 12783 是一種特異性，有效且選擇性的多巴胺攝取抑制劑，可抑制大鼠和小鼠紋狀體突觸小體對 [3H] 多巴胺 ([3H]dopamine) 的攝取，IC50 分別為 1.8 nM 和 1.2 nM。GBR 12783 還可改善大鼠記憶力并增加海馬通路乙酰膽堿的釋放。

Eldecalcitol (ED-71) 是1,25-二羥基維生素D3的類似物。

LDE-225 HCl是有效，選擇性的 Smo 拮抗劑， 抑制鼠和人Smo的 IC50 分別為 1.3 nM 和 2.5 nM。

Oseltamivir phosphate (GS 4104) 是一種神經氨酸酶 (neuraminidase) 抑制劑，用于預防和治療流感 (influenza A 和 B)。

Deferasirox (ICL 670) 是具有口活性的，用于治療鐵離子過量的螯合劑。

Peramivir trihydrate (RWJ-270201 trihydrate;BCX-1812 trihydrate) 是一種高效、選擇性和口服有效的流感病毒神經氨酸酶 (NA) 抑制劑，對 9 個亞型 NA 抑制作用的 IC50 值為 0.9-4.3 nM。

Ibudilast(KC-404;AV-411;MN-166) is a relatively nonselective phosphodiesterase inhibitor which has been marketed for treating asthma,ibudilast (MN-166) is tested to treat acute respiratory distress syndrome (ARDS) associated with Covid-19.

Paroxetine hydrochloride hemihydrate is a antidepressant agents known as selective serotonin-reuptake inhibitors (SSRIs).

Tamoxifen(ICI-46474) is an antagonist of the estrogen receptor in breast tissue via its active metabolite, hydroxytamoxifen,showed potent activity against COVID-19(SARS-COV-2) with EC50 MERS-COV(10.117), SARS-COV(11.696).

Clevudine (Levovir) is an antiviral drug for the treatment of hepatitis B,showed potent activity against COVID-19(SARS-COV-2) .

Ribavirin is a guanosine analog with antiviral properties against DNA and RNA viruses, including respiratory syncytial virus, hepatitis C, and influenza.

Atovaquone is a medication used to treat or prevent for pneumocystis pneumonia, toxoplasmosis, malaria, and babesia.

Darunavir(TMC114) is an HIV protease inhibitor,showed potent activity against COVID-19(SARS-COV-2) .

Felbamate (Felbatol) is an anticonvulsant drug used in the treatment of epilepsy.

6-Thioguanine(6-TG) belongs to the thiopurine family of drugs that also include mercaptopurine and azathioprine, which are examples of antimetabolites; it is a purine analogue of the nucleobase guanine.

Gabapentin (Neurontin) is a pharmaceutical drug, specifically a GABA analog. It was originally developed to treat epilepsy, and currently is also used to relieve neuropathic pain.

Carmustine is a cell-cycle phase nonspecific alkylating antineoplastic agent.

Riluzole is a glutamate antagonist used as an anticonvulsant and to prolong the survival of patients with amyotrophic lateral sclerosis.

Imiquimod is an immune response modifier that acts as a toll-like receptor 7 agonist and is commonly used topically to treat warts on the skin of the genital and anal areas.

Triamterene blocks epithelial Na+ channel (ENaC) in a voltage-dependent manner, which used as a mild diuretic.

Cyclophosphamide is a synthetic alkylating agent chemically related to the nitrogen mustards with antineoplastic and immunosuppressive activities.